Drug × Cancer matrix

Each row is a drug, each column a cancer subtype. Cells show the strongest known association for that drug in that cancer: approved clinical trial or blank. The repositionable flag means the drug appears as a synthetic-lethal repositioning candidate in cansar; it’s gene-level, not cancer-level.

Cancer key
GBM — Glioblastoma (CNS astrocytoma grade IV) LUAD — Lung adenocarcinoma SCLC — Small cell lung carcinoma LUSC — Lung squamous cell carcinoma OAC — Oesophageal adenocarcinoma OSCC — Oesophageal squamous cell carcinoma PDAC — Pancreatic ductal adenocarcinoma
Clear
Showing 68 of 68 matching drugs for CSF3R — including drugs targeting any of its 23 synthetic-lethal partners , sorted by total cancer coverage.
Drug Target Relationship GBM LUAD SCLC LUSC OAC OSCC PDAC Reposition #cancers
filgrastim, paclitaxel, topotecan hydrochloride CSF3R Direct 2
aldesleukin, autologous tumor cell vaccine, filgrastim, sargramostim, therapeutic autologous lymphocytes, carmustine, cisplatin, cyclophosphamide, paclitaxel, autologous bone marrow transplantation, conventional surgery, peripheral blood stem cell transplantation CSF3R Direct 1
anti-thymocyte globulin, filgrastim, busulfan, cyclophosphamide, cyclosporine, fludarabine phosphate, melphalan, methylprednisolone, umbilical cord blood transplantation, radiation therapy CSF3R Direct 1
anti-thymocyte globulin, filgrastim, busulfan, cyclophosphamide, methylprednisolone, umbilical cord blood transplantation, radiation therapy CSF3R Direct 1
cetuximab, filgrastim, fluorouracil, irinotecan hydrochloride, leucovorin calcium CSF3R Direct 1
epoetin alfa, filgrastim, cisplatin, fluorouracil, gemcitabine hydrochloride, adjuvant therapy, conventional surgery, neoadjuvant therapy, radiation therapy CSF3R Direct 1
filgrastim, amifostine trihydrate, cisplatin, etoposide, paclitaxel, topotecan hydrochloride, radiation therapy CSF3R Direct 1
filgrastim, busulfan, cyclophosphamide, etoposide, melphalan, autologous-autologous tandem hematopoietic stem cell transplantation, radiation therapy CSF3R Direct 1
filgrastim, carboplatin, cisplatin, cyclophosphamide, etoposide, thiotepa, vincristine sulfate, conventional surgery, peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, carboplatin, cyclophosphamide, etoposide, autologous bone marrow transplantation, peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, carboplatin, cyclophosphamide, paclitaxel, topotecan hydrochloride, peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, carboplatin, etoposide, bone marrow ablation with stem cell support, peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, carboplatin, etoposide, ifosfamide, in vitro-treated peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, carboplatin, etoposide, isotretinoin, thiotepa, autologous bone marrow transplantation, peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, carboplatin, etoposide, paclitaxel, topotecan hydrochloride, radiation therapy CSF3R Direct 1
filgrastim, carboplatin, paclitaxel, topotecan hydrochloride CSF3R Direct 1
filgrastim, carboplatin, temozolomide, thiotepa, autologous bone marrow transplantation, peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, carboplatin, thiotepa, autologous bone marrow transplantation, peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, cisplatin, fluorouracil, paclitaxel, radiation therapy CSF3R Direct 1
filgrastim, docetaxel, gemcitabine hydrochloride CSF3R Direct 1
filgrastim, exatecan mesylate CSF3R Direct 1
filgrastim, gemcitabine hydrochloride, vinorelbine tartrate CSF3R Direct 1
filgrastim, gene therapy, lomustine, procarbazine hydrochloride, vincristine sulfate, in vitro-treated peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, pegfilgrastim, cisplatin, fluorouracil, paclitaxel, conventional surgery, radiation therapy CSF3R Direct 1
filgrastim, recombinant interferon alfa, fluorouracil, hydroxyurea CSF3R Direct 1
filgrastim, sargramostim, cyclophosphamide, thiotepa, autologous bone marrow transplantation, bone marrow ablation with stem cell support, peripheral blood stem cell transplantation CSF3R Direct 1
filgrastim, temozolomide, peripheral blood stem cell transplantation CSF3R Direct 1
fludarabine phosphate, cyclophosphamide, rituxan (rituximab), filgrastim, methylprednisolone, immunologic technique, laboratory biomarker analysis, autologous hematopoietic stem cell transplantation, diphenhydramine, mesna CSF3R Direct 1
gemcitabine, ribociclib, sonidegib, trametinib, filgrastim CSF3R Direct 1
laboratory biomarker analysis, pegfilgrastim, pharmacological study, tivantinib, topotecan hydrochloride CSF3R Direct 1
ly2523355, pegfilgrastim CSF3R Direct 1
o6-benzylguanine, temozolomide, filgrastim, pharmacological study, laboratory biomarker analysis CSF3R Direct 1
p140k-mgmt, o6-benzylguanine, photon based radiotherapy, temozolomide, filgrastim, carmustine CSF3R Direct 1
filgrastim CSF3R Direct yes 0
pegfilgrastim CSF3R Direct yes 0
unnamed compound CSF3R Direct yes 0
adjuvant therapy, temozolomide, valproic acid, radiation therapy CDKN1A SSL via CDKN1A 1
adriamycin, cyclophosphamide, vindesine, valproic acid CDKN1A SSL via CDKN1A 1
arsenic trioxide CDKN1A SSL via CDKN1A 1
arsenic trioxide, radiation therapy CDKN1A SSL via CDKN1A 1
arsenic trioxide, temozolomide, adjuvant therapy, intensity-modulated radiation therapy, radiation therapy CDKN1A SSL via CDKN1A 1
atorvastatin, temozolomide, radiotherapy HMGCR SSL via HMGCR 1
irinotecan, cisplatin, simvastatin HMGCR SSL via HMGCR 1
medical cannabis HMGCR SSL via HMGCR 1
nabiximols, temozolomide, nabiximols-matched placebo HMGCR SSL via HMGCR 1
rosuvastatin HMGCR SSL via HMGCR yes 1
sorafenib tosylate, valproic acid, sildenafil citrate CDKN1A SSL via CDKN1A 1
valproic acid CDKN1A SSL via CDKN1A 1
valproic acid, bevacizumab, radiation therapy CDKN1A SSL via CDKN1A 1
valproic acid, simvastatin 20mg, gemcitabine 1000 mg, nab paclitaxel, cisplatin, capecitabine CDKN1A SSL via CDKN1A 1
atorvastatin HMGCR SSL via HMGCR yes 0
atorvastatin calcium HMGCR SSL via HMGCR yes 0
cerivastatin HMGCR SSL via HMGCR yes 0
cerivastatin sodium HMGCR SSL via HMGCR yes 0
fluvastatin HMGCR SSL via HMGCR yes 0
fluvastatin sodium HMGCR SSL via HMGCR yes 0
lemborexant HCRTR1 SSL via HCRTR1 yes 0
lovastatin HMGCR SSL via HMGCR yes 0
midostaurin PRKCD SSL via PRKCD yes 0
pitavastatin HMGCR SSL via HMGCR yes 0
pitavastatin calcium HMGCR SSL via HMGCR yes 0
pitavastatin magnesium HMGCR SSL via HMGCR yes 0
pitavastatin sodium HMGCR SSL via HMGCR yes 0
pravastatin HMGCR SSL via HMGCR yes 0
pravastatin sodium HMGCR SSL via HMGCR yes 0
rosuvastatin calcium HMGCR SSL via HMGCR yes 0
simvastatin HMGCR SSL via HMGCR yes 0
suvorexant HCRTR1 SSL via HCRTR1 yes 0
Approval data manually curated from National Cancer Institute and Drugs@FDA. Clinical trials from ClinicalTrials.gov. Repositionable list from cansar.ai.