ADRA1A

Alpha-1D adrenergic receptor UniProt accession P25100

Alpha-1 adrenergic receptors are G protein-coupled receptors for catecholamines that signal through the G(q) family of G proteins, including G(q) and G(11). Upon activation, they stimulate the phosphatidylinositol-calcium second messenger pathway, leading to calcium release from intracellular stores and activation of protein kinase C (PubMed:7746284). ADRA1D binds the catecholamine ligands norepinephrine and epinephrine (PubMed:7815325, PubMed:8024574, PubMed:8183249)

Source: UniProt

Interacts with FLNA (via filamin repeat 21); increases PKA-mediated phosphorylation of FLNA

Source: UniProt
Cell membrane — Multi-pass membrane protein
Source: UniProt
  • Adrenoceptors
  • G alpha (q) signalling events
  • G alpha (12/13) signalling events
Source: Reactome via UniProt

Mutations

No mutation information available.

Synthetic Lethal Network

Genes with an experimentally identified or computationally predicted synthetic-lethal relationship to ADRA1A, aggregated across our SSL data sources. Click any partner node to view that gene’s page.

Nodes and edges are coloured by the SSL data source. Partners appearing in more than one source are shown in grey.

BioGRID SLOrth SynLethDB MexDrugs Multi-source
Sources: BioGRID, SLOrth, SynLethDB, MexDrugs

Clinical Trials

Total Trials Found: 1

NCT ID Condition Brief Title Phase Status
NCT03132272 Alzheimer Dementia Immunoadsorption for Treatment of Alzheimer's Disease NA TERMINATED