PPARD

Peroxisome proliferator-activated receptor delta UniProt accession Q03181

Ligand-activated transcription factor key mediator of energy metabolism in adipose tissues (PubMed:35675826). Receptor that binds peroxisome proliferators such as hypolipidemic drugs and fatty acids. Has a preference for poly-unsaturated fatty acids, such as gamma-linoleic acid and eicosapentanoic acid.

Once activated by a ligand, the receptor binds to promoter elements of target genes. Regulates the peroxisomal beta-oxidation pathway of fatty acids. Functions as transcription activator for the acyl-CoA oxidase gene.

Decreases expression of NPC1L1 once activated by a ligand

Source: UniProt

Heterodimer with the retinoid X receptor. Interacts (via domain NR LBD) with CRY1 and CRY2 in a ligand-dependent manner (By similarity)

Source: UniProt
Nucleus
Source: UniProt

Ubiquitous with maximal levels in placenta and skeletal muscle

Source: UniProt
  • Carnitine shuttle
  • Nuclear Receptor transcription pathway
  • Signaling by Retinoic Acid
Source: Reactome via UniProt

Mutations

No mutation information available.

Synthetic Lethal Network

Genes with an experimentally identified or computationally predicted synthetic-lethal relationship to PPARD, aggregated across our SSL data sources. Click any partner node to view that gene’s page.

Nodes and edges are coloured by the SSL data source. Partners appearing in more than one source are shown in grey.

BioGRID SLOrth SynLethDB MexDrugs Multi-source
Sources: BioGRID, SLOrth, SynLethDB, MexDrugs

Clinical Trials

Total Trials Found: 3

NCT ID Condition Brief Title Phase Status
NCT00841217 Obesity, Lipid Disorders, Cardiovascular Disease Regulation of Lipoprotein Transport in Metabolic Syndrome PHASE4 COMPLETED